Tag: tropane

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106. Synthesis of 2β-Acyl-3β-(substituted naphthyl)-8-azabicyclo[3.2.1]octanes and Their Binding Affinities at Dopamine and Serotonin Transport Sites

Authors: Huw M. L. Davies , Vernon Gilliatt , Lisa A. Kuhn , Elie Saikali , Pingda Ren , Philip S. Hammond , Tammy Sexton  and Steven R. Childers

J. Med. Chem.,

2001, 44 (10), 1509–1515

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103. A cocaine analog, 2β-propanoyl-3β-(4-tolyl)-tropane (PTT), reduces tyrosine hydroxylase in the mesolimbic dopamine pathway

Authors: Willard M Freeman, George J Yohrling IV, James B Daunais, Lynda Gioia, Stephanie L Hart, Linda J Porrino, Huw M.L Davies, Kent E Vrana

Drug and Alcohol Dependence

2000, 61, 1, 15-21

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93. Characterization of a Tropane Radioligand, [3H]2β-Propanoyl-3β-(4-tolyl) Tropane ([3H]PTT), for Dopamine Transport Sites in Rat Brain

Authors: Sharon R. Letchworth, Hilary R. Smith, Linda J. Porrino, Barbara A. Bennett, Huw M. L. Davies, Tammy Sexton and Steven R. Childers

J. Pharmacol. Exp. Therap.,

2000, 293, 2, 686-696

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105. Synthesis and monoamine transporter affinity of 3β-(4-(2-pyrrolyl)phenyl)-8-azabicyclo[3.2.1]octanes and 3β-(5-Indolyl)-8-azabicyclo[3.2.1]octanes

Authors: Huw M.L Davies, Pingda Ren, Norman Kong, Tammy Sexton, Steven R Childers

Bioorganic & Medicinal Chemistry Letters

2001, 11, 4, 487-489

Continue reading “105. Synthesis and monoamine transporter affinity of 3β-(4-(2-pyrrolyl)phenyl)-8-azabicyclo[3.2.1]octanes and 3β-(5-Indolyl)-8-azabicyclo[3.2.1]octanes”